| 名称
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Luteinizing Hormone-Releasing Hormone Anta
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| 编码
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[292141-31-2]
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| 别名
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Luteinizing Hormone-Releasing Hormone Anta
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| 纯度
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80%，90%，95%，98%，99%
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| 重量
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1mg,5mg,10mg,50mg,100mg,1g
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| 序列（单字母缩写）
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Ac-D-2-Nal-p-chloro-f-beta-(3-pyridyl)-AGRPa-NH2
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| 序列（三字母缩写）
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Ac-D-2-Nal-p-chloro-D-Phe-beta-(3-pyridyl)-D-Ala-Gly-Arg-Pro-D-Ala-NH2?(trifluoroacetate salt)
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| 基本描述
|
GnRH antagonist. CAS Number (cetrorelix acetate): 145672-81-7. This peptide is offered and sold solely for uses reasonably related to the development and submission of information under a Federal law which regulates the manufacture, use or sale of drugs (the ?Bolar Exemption?). Bachem cannot be made liable for any infringement of intellectual property rights. It is the sole and only responsibility of the purchaser or user of this product to comply with the relevant national rules and regulations. A highly modified luteinizing hormone-releasing hormone (LHRH) decapeptide with a terminal amide group, this peptide is a LHRH antagonist. It regulates the expression of Galphas and Galphai protein subunits and adenylate cyclase activity in ovary, breast and pituitary. Cetrorelix competitively inhibits LHRH receptor in the pituitary gland to suppress ovarian and testicular functions.
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| 溶解度
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| 分子量
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967.53
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| 化学式
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C48H59Cl1N12O8
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| 存储条件
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Store at -20°C. Keep tightly closed. Store in a cool dry place.
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| 注释
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| Documents
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| Figures
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| Reference
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D.Yahalom et al., J. Med. Chem., 43, 2831 (2000)
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| 化学桥
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